Nenitzescu吲哚合成反应

对苯醌和β-胺基巴豆酸酯缩合得到5-羟基吲哚的反应。

反应机理

反应实例

参考文献

1. Nenitzescu, C. D. Bull. Soc. Chim. Romania 1929, 11, 37-􀀐43.

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Sheinker, Y. N.; Granik, V. G. Tetrahedron 1997, 53, 177􀀐-184.

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9. Li, J.; Cook, J. M. Nenitzescu indole synthesis. In Name Reactions in Heterocyclic Chemistry; Li, J. J., Ed.; Wiley: Hoboken, NJ, 2005, pp 145􀀐-153. (Review).

10. Velezheva, V. S.; Sokolov, A. I.; Kornienko, A. G.; Lyssenko, K. A.; Nelyubina, Y.V.; Godovikov, I. A.; Peregudov, A. S.; Mironov, A. F. Tetrahedron Lett. 2008, 49,7106-􀀐7109.

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编译自：Name Reactions （A Collection of Detailed Reaction Mechanisms）, Jie Jack Li, Nenitzescu indole synthesis，page 432-433.